Characteristics
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Cell-permeable. A potent, non-competitive inhibitor of p300 and PCAF (p300/CBP-associated factor) histone acetyltransferase (HAT) activities (IC50 approx. 8.5 µM and approx. 5 µM, respectively. Inhibits SUMOylation of RanGAP1-C2with an IC50 = 2.2 µM
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