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  • 产品名称:PI3-KɣInhibitor,AS-605240

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简单介绍:
PI3-KɣInhibitor,AS-605240
详情介绍:
Purpose A potent inhibitor of PI 3-kinase γ (PI3Kγ)
Characteristics A potent and selective inhibitor of PI 3-kinase gamma (PI3Kgamma) (IC50 = 8 nM). Displays >33-fold selectivity over PI3Kdelta and PI3Kbeta and 7.5-fold selectivity over PI3Kalpha.
Purity ≥ 98 % by HPLC
Chemical Name 5-(6-Quinoxalinylmethylene)-2,4-thiazolidine-2,4-dione
Formula C₁₂H₇N₃O₂S
Permeability Cell-permeable
Solubility DMSO ( 1 mM)
Molecular Weight 257.27 g/mol
CAS-No 648450-29-7
Research Area Kinases/Phosphatases
Restrictions For Research Use only
Format Solid
Handling Advice Protect from air and light
Storage -20 °C
Expiry Date 48 months
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